SCHEMBL6676181

SCHEMBL6676181

NCCc1ccc(N)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.56
CYP3A4 P08684 4/20 0.52
TSHR P16473 2/20 0.52
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
PNMT P11086 1/20 0.43
MAOB P27338 2/20 0.41
ALDH1A1 P00352 3/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
EPHX2 P34913 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
PDE7A Q13946 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1299722 0.86 CYP3A4 (0.52) TAAR1CYP3A4TSHRCA1CA2
SCHEMBL14085077 0.84 CYP3A4 (0.54) CYP3A4TSHRCA1CA2PNMT
SCHEMBL3787093 0.83 CYP3A4 (0.48) TAAR1CYP3A4TSHRCA1CA2
SCHEMBL11292184 0.83 CYP3A4 (0.48) TAAR1CYP3A4TSHRCA1CA2
SCHEMBL29362177 0.83 CA1 (0.48) TAAR1CYP3A4TSHRCA1CA2
SCHEMBL1625228 0.83 CA1 (0.48) TAAR1CYP3A4TSHRCA1CA2
SCHEMBL473578 0.82 IDO1 (0.56) TAAR1CYP3A4TSHRMAOB
SCHEMBL29787088 0.82 IDO1 (0.56) TAAR1CYP3A4TSHRMAOB
SCHEMBL31175763 0.81 CYP3A4 (0.56) CYP3A4TSHRCA1CA2ALDH1A1
SCHEMBL352023 0.81 CYP3A4 (0.56) CYP3A4TSHRCA1CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113979893-B N-hydroxy formamidine derivative, preparation method and application 中国药科大学 2023-10-24 CN disclosed
CN-113979893-A N-hydroxyformamidine derivative, preparation method and application 中国药科大学 2022-01-28 CN disclosed
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
CN-1075808-C Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-12-05 CN disclosed
CN-1310169-A Anils with nitric oxide synzyme inhibiting function SHUGAI SEIYAKU K K (JP) 2001-08-29 CN disclosed
CN-1172473-A Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-02-04 CN disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed