SCHEMBL6679160

SCHEMBL6679160

COC(=O)c1cc(N=C(NO)N2CCN(c3cc(OC)cc(OC)c3)CC2)c(OC)nc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
GAA P10253 3/20 0.39
KMT2A Q03164 7/20 0.38
MAPT P10636 3/20 0.38
MAPK1 P28482 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GFER P55789 1/20 0.37
CCKAR P32238 1/20 0.36
PKM P14618 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675909 0.92 PHGDH (0.40) PHGDHGAAKMT2AMAPTMAPK1
SCHEMBL6676074 0.91 GAA (0.40) PHGDHCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6673384 0.90 GAA (0.39) CYP2C9CYP2C19GAAKMT2AMAPT
SCHEMBL6675492 0.90 MAPT (0.45) CYP2C9CYP2C19CYP1A2CYP3A4GAA
SCHEMBL6673176 0.90 GAA (0.39) CYP2C9CYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL6679148 0.88 KMT2A (0.37) PHGDHCYP2C9CYP2C19GAAKMT2A
SCHEMBL6673426 0.88 PHGDH (0.39) PHGDHCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6673102 0.87 KDM4E (0.46) KMT2AMAPTL3MBTL1SMN1; SMN2MEN1
SCHEMBL6672608 0.87 PHGDH (0.43) PHGDHCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6678302 0.85 PHGDH (0.40) PHGDHGAAKMT2AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1424072-A1 N'-(pyridin-3-yl)-(4-phenylpiperazin-1-yl)-carboxyimidamide and -iminothiolate derivatives for the treatment of tumors Samjin Pharmaceutical Co., Ltd. (KR) 2004-06-02 EP disclosed
US-6683184-B2 ANTITUMOR AGENTS SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2004-01-27 US disclosed