SCHEMBL6682278

SCHEMBL6682278

CCNC(=NC(=O)OC(C)(C)C)Nc1ccc(N2CCCC2)c(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
RECQL P46063 2/20 0.39
ALDH1A1 P00352 4/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 1/20 0.36
MAPT P10636 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
HTT P42858 1/20 0.33
GAA P10253 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
NR1I3 Q14994 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679942 0.87 MCHR1 (0.32) BACE1HTT
SCHEMBL6675981 0.86 CNR2 (0.33) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL6678082 0.85 HTT (0.35) ALDH1A1KMT2AMEN1CYP2D6CYP2C19
SCHEMBL6675631 0.85 GRM2 (0.35) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL6681137 0.85 MCHR1 (0.31)
SCHEMBL6675983 0.85 NR1H4 (0.33)
SCHEMBL6679125 0.85 MCHR1 (0.31)
SCHEMBL6679306 0.84 KDM4E (0.43) KDM4ERECQLALDH1A1KMT2AMEN1
SCHEMBL6684398 0.83 MCHR1 (0.32)
SCHEMBL6686111 0.82 MCHR1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed