SCHEMBL6683563

SCHEMBL6683563

CC(CCCBr)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
IDO1 P14902 2/20 0.36
TDO2 P48775 2/20 0.36
MC4R P32245 3/20 0.34
TSHR P16473 1/20 0.33
CYP19A1 P11511 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
HIF1A Q16665 1/20 0.32
CNR2 P34972 1/20 0.32
ACHE P22303 1/20 0.31
PKM P14618 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7562080 0.93 CYP3A4 (0.35) CYP3A4IDO1TDO2MC4RTSHR
SCHEMBL17858417 0.89 CYP3A4 (0.38) CYP3A4IDO1TDO2MC4RTSHR
SCHEMBL20710583 0.83 HRH1 (0.44) CYP3A4IDO1TDO2TSHRCYP19A1
SCHEMBL9286802 0.83 TSHR (0.38) CYP3A4IDO1TDO2MC4RTSHR
SCHEMBL9229150 0.83 TSHR (0.38) CYP3A4IDO1TDO2MC4RTSHR
SCHEMBL19215837 0.81 CYP3A4 (0.36) CYP3A4IDO1TDO2TSHRCYP19A1
SCHEMBL15022607 0.81 CYP3A4 (0.40) CYP3A4IDO1TDO2TSHRALDH1A1
SCHEMBL24920008 0.80 CSNK1E (0.41) CYP3A4TSHRALDH1A1MEN1KMT2A
SCHEMBL5795839 0.79 HTT (0.39) CYP3A4IDO1TDO2TSHRALDH1A1
SCHEMBL18007088 0.79 ESR1 (0.41) CYP3A4MC4RTSHRCYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111056-A2 COMPOUND LIBRARIES OF SPIRO-BENZODIOXINE-PIPERIDINES BIOFOCUS PLC (GB) 2004-12-23 WO disclosed
WO-2004035568-A1 BENZOFURAN DERIVATIVES, FORMULATIONS AND USES THEREOF UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 2004-04-29 WO disclosed