SCHEMBL6685301

SCHEMBL6685301

Cc1nc(C(=O)N2CCCC[C@@H]2CC(=O)OCC(=O)c2ccccc2F)c(-c2ccc(F)cc2)s1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.60
HCRTR2 O43614 15/20 0.60
TSPO P30536 1/20 0.47
OPRK1 P41145 1/20 0.47
HTR2B P41595 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1778604 1.00 HCRTR1 (0.60) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL1777548 0.92 HCRTR1 (0.60) HCRTR1HCRTR2
SCHEMBL1778797 0.92 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL1779324 0.92 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL1778624 0.91 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL6692756 0.91 HCRTR1 (0.64) HCRTR1HCRTR2
SCHEMBL1777329 0.90 HCRTR1 (0.60) HCRTR1HCRTR2
SCHEMBL1780233 0.87 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL1780504 0.85 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL1256951 0.84 HCRTR1 (0.66) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406897-A2 COMPOUNDS SmithKline Beecham plc (GB) 2004-04-14 EP disclosed
WO-2003002559-A2 PIPERIDINE COMPOUNDS FOR USE AS OREXIN RECEPTOR ANTAGONIST SMITHKLINE BEECHAM P.L.C. (GB) 2003-01-09 WO disclosed