SCHEMBL6687151

SCHEMBL6687151

O=C(Nc1nc2ccccc2s1)c1ccc(-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 7/20 1.00
NPC1 O15118 4/20 0.83
RAB9A P51151 4/20 0.83
MEN1 O00255 3/20 0.83
KMT2A Q03164 3/20 0.83
SMN1; SMN2 Q16637 2/20 0.83
KDM4E B2RXH2 3/20 0.75
HTT P42858 2/20 0.75
NFKB1 P19838 1/20 0.75
NFKB2 Q00653 1/20 0.75
RELA Q04206 1/20 0.75
MMP13 P45452 1/20 0.68
TOP1 P11387 2/20 0.67
CASP3 P42574 1/20 0.65
SENP8 Q96LD8 1/20 0.65
SENP7 Q9BQF6 1/20 0.65
SENP6 Q9GZR1 1/20 0.65
LRRK2 Q5S007 2/20 0.62
CSNK1D P48730 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3053529 0.91 NPC1 (1.00) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL16562172 0.90 NPC1 (0.86) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL17916702 0.89 SCD (1.00) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL2754053 0.87 SCD (0.93) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL19464549 0.86 NPC1 (0.79) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL16562119 0.86 NPC1 (0.80) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL4910843 0.86 NPC1 (0.78) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL4920257 0.86 NPC1 (0.78) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL30553332 0.86 NPC1 (0.78) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL4917567 0.86 NPC1 (1.00) SCDNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078115-A2 BENZOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT AND PROPHYLAXIS OF ROTAVIRUS INFECTIONS AND ASSOCIATED DISEASES VIROPHARMA, INCORPORATED (US) 2004-09-16 WO claimed
US-9789096-B2 Methods and compositions for selective and targeted cancer therapy BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-10-17 US disclosed
US-9789096-B2 Methods and compositions for selective and targeted cancer therapy BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-10-17 US disclosed
US-20160200695-A1 Methods and Compositions for Selective and Targeted Cancer Therapy BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-07-14 US disclosed
US-20160200695-A1 Methods and Compositions for Selective and Targeted Cancer Therapy BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-07-14 US disclosed
WO-2015035051-A1 METHODS AND COMPOSITIONS FOR SELECTIVE AND TARGETED CANCER THERAPY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-03-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160200695-A1 Methods and Compositions for Selective and Targeted Cancer Therapy NCOA4, SREBF1, ACOX1 SCD 4/4885NPC1 840/4885RAB9A 4781/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.