SCHEMBL6689772

SCHEMBL6689772

O=C(O)c1ccc2c(c1)S(=O)(=O)N=C(c1c(O)c3cc(F)ccc3n(CCC3CC3)c1=O)N2

nearest known ligand 0.78

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.78
NR1I2 O75469 1/20 0.78
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PLK1 P53350 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
PTGER4 P35408 1/20 0.36
KDM4C Q9H3R0 1/20 0.34
CA12 O43570 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
HTR2A P28223 1/20 0.34
DRD3 P35462 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687473 0.93 CYP2C9 (0.77) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6687698 0.91 CYP2C9 (0.72) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6733802 0.91 CYP2C9 (0.77) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6689094 0.91 CYP2C9 (0.76) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6690316 0.90 CYP2C9 (0.83) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6209607 0.90 CYP2C9 (0.66) CYP2C9NR1I2MAPK1HSD17B10PTGER4
SCHEMBL6693468 0.90 CYP2C9 (0.81) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6232054 0.89 CYP2C9 (0.80) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL5089690 0.88 CYP2C9 (1.00) CYP2C9NR1I2MAPK1HSD17B10PLK1
SCHEMBL6687474 0.88 CYP2C9 (0.69) CYP2C9NR1I2MAPK1HSD17B10PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052313-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO disclosed