SCHEMBL6691669

SCHEMBL6691669

CCOc1ccc(C(CC(=O)O)N2C(=O)c3cccc(N)c3C2=O)cc1OCC

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 15/20 0.71
PDE4B Q07343 15/20 0.71
PDE4C Q08493 15/20 0.71
PDE4D Q08499 15/20 0.71
TNF P01375 5/20 0.67
HTR2B P41595 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21494489 0.95 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL23000612 0.95 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL21494487 0.95 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6693901 0.92 TNF (0.80) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6692793 0.88 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL537289 0.88 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL537150 0.88 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6690298 0.88 TNF (0.83) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL3128437 0.87 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL21494520 0.86 TNF (0.87) PDE4APDE4BPDE4CPDE4DTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1477486-A2 Imides as inhibitors of TNF alpha CELGENE CORPORATION (US) 2004-11-17 EP claimed
EP-0706521-B1 IMIDES AS TNF ALPHA INHIBITORS CELGENE CORP (US) 2002-10-02 EP claimed
WO-2019201255-A1 ISOINDOLE DERIVATIVE 天津合美医药科技有限公司 2019-10-24 WO disclosed