SCHEMBL6711441

SCHEMBL6711441

O=C1C(NS(=O)(=O)c2cc3nc(Cl)ccc3s2)CCCN1c1ccc(-n2ccccc2=O)cc1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F10 P00742 20/20 0.78
F2 P00734 3/20 0.50
PLG P00747 3/20 0.50
PROC P04070 2/20 0.50
PRSS1 P07477 2/20 0.50
PLAT P00750 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5619613 0.87 F10 (1.00) F10
SCHEMBL6712834 0.81 F10 (0.69) F10F2
SCHEMBL4479220 0.78 F10 (1.00) F10
SCHEMBL4477449 0.78 F10 (0.81) F10F2PLGPROCPRSS1
SCHEMBL4484131 0.76 F10 (0.65) F10
SCHEMBL4472147 0.76 F10 (0.80) F10
SCHEMBL14603100 0.75 F10 (0.63) F10F2PLGPROCPRSS1
SCHEMBL6714527 0.74 F10 (0.75) F10
SCHEMBL14603293 0.73 F10 (0.77) F10F2PLGPROCPRSS1
SCHEMBL14337591 0.73 F10 (0.57) F10F2PLGPROCPRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040006062-A1 Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040006062-A1 Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors TFPI, SPINT2, PRSS1 F10 31/4885F2 21/4885PLG 25/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.