SCHEMBL6723798

SCHEMBL6723798

C[Si](C)(C)CCOCn1c(=O)[nH]c(=O)c2cccnc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
KDM4D Q6B0I6 2/20 0.40
CYP1A2 P05177 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
HCAR2 Q8TDS4 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
LDHA P00338 1/20 0.36
MAPT P10636 1/20 0.36
EGFR P00533 1/20 0.36
IGF1R P08069 1/20 0.36
SRC P12931 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
FLT3 P36888 1/20 0.36
EPHB4 P54760 1/20 0.36
TEK Q02763 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6723898 0.81 PNP (0.36) NPC1ALDH1A1HPGDMAPT
SCHEMBL6719104 0.81 NPC1 (0.53) NPC1CYP1A2CYP2C9ALDH1A1HPGD
SCHEMBL6722467 0.74 PDE4A (0.60) CYP1A2ALDH1A1
SCHEMBL17967647 0.74 MAPT (0.44) NPC1POLBPKMCYP1A2CYP2C9
Ammonia Solution, Strong SCHEMBL27784212 0.73 NPC1 (0.38) NPC1POLBPKMMAPT
SCHEMBL30046010 0.73 NPC1 (0.45) NPC1MAPTEGFRSRC
SCHEMBL555692 0.73 BRD4 (0.60) POLBALDH1A1
SCHEMBL6726785 0.72 NPC1 (0.37) NPC1ALDH1A1MAPTEGFRIGF1R
SCHEMBL29674632 0.72 NPC1 (0.46) NPC1POLBPKMALDH1A1MAPT
SCHEMBL25246336 0.72 NPC1 (0.34) NPC1POLBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673804-B1 PREVENTING OR TREATING ARTHRITIS (PARTICULARLY OSTEOARTHRITIS) OR INHIBITING METASTASIS, INVASION OR GROWTH OF CANCER (PARTICULARLY BREAST CANCER) SANKYO COMPANY, LIMITED (JP) 2004-01-06 US disclosed
EP-1069110-A1 SULFONAMIDE DERIVATIVES Sankyo Company Limited (JP) 2001-01-17 EP disclosed