SCHEMBL673107

SCHEMBL673107

CCc1noc(C(C)N(c2cc(C#CC(C)(C)C)sc2C(=O)O)C(=O)[C@H]2CC[C@H](C)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.54
NR1I2 O75469 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10205786 1.00 CYP2E1 (0.54) CYP2E1NR1I2
SCHEMBL15498384 0.92 CYP2E1 (0.45) CYP2E1NR1I2
SCHEMBL15511997 0.92 CYP2E1 (0.45) CYP2E1NR1I2
SCHEMBL15498381 0.91 CYP2E1 (0.55) CYP2E1NR1I2
SCHEMBL15498383 0.85 CYP2E1 (0.61) CYP2E1NR1I2
SCHEMBL15498302 0.85 CYP2E1 (0.61) CYP2E1NR1I2
SCHEMBL15498382 0.83 CYP2E1 (0.46) CYP2E1NR1I2
SCHEMBL670676 0.83 CYP2E1 (0.46) CYP2E1NR1I2
SCHEMBL14718058 0.82 NR1I2 (0.61) CYP2E1NR1I2
SCHEMBL102096 0.82 NR1I2 (0.61) CYP2E1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606041-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRIDAE VIRAL INFECTIONS Vertex Pharmaceuticals Incorporated (US) 2013-06-26 EP disclosed
WO-2012024363-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRIDAE VIRAL INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-23 WO disclosed