SCHEMBL6747697

SCHEMBL6747697

CCCCc1ccc(S(=O)(=O)Nc2nccnc2-c2ccc(-n3c(CC)nc4ccccc43)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 10/20 0.55
BACE1 P56817 1/20 0.45
KIT P10721 1/20 0.41
KDM4E B2RXH2 1/20 0.39
EDNRA P25101 1/20 0.39
FAAH O00519 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NTRK1 P04629 1/20 0.38
NTRK2 Q16620 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6751658 0.77 PTGDR2 (0.53) PTGDR2BACE1KITKDM4E
SCHEMBL6751309 0.73 PTGDR2 (0.47) PTGDR2BACE1KITALDH1A1MEN1
SCHEMBL2442871 0.71 PTGDR2 (1.00) PTGDR2EDNRA
SCHEMBL1624962 0.69 PTGER4 (0.71) ALDH1A1MAPTCYP2C9NTRK1NTRK2
SCHEMBL2444077 0.69 PTGDR2 (1.00) PTGDR2
SCHEMBL1625482 0.67 RECQL (0.51) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL1624977 0.67 NTRK1 (0.52) KDM4EFAAHALDH1A1MEN1KMT2A
SCHEMBL2449413 0.66 PTGDR2 (0.57) PTGDR2ALDH1A1
SCHEMBL12402570 0.65 BACE1 (0.82) BACE1KDM4EALDH1A1MEN1KMT2A
SCHEMBL3948783 0.65 NTRK1 (0.48) KDM4EALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058265-A1 COMPOUND LIBRARIES OF 2,3-SUBSTITUTED PYRAZINE DERIVATIVES CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed