SCHEMBL6749588

SCHEMBL6749588

COc1cccc(OCc2ccc(-c3nccnc3C#N)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.53
APP P05067 1/20 0.52
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SMPD1 P17405 1/20 0.42
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
NAAA Q02083 1/20 0.41
FFAR1 O14842 2/20 0.41
ADAMTS4 O75173 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2056993 0.82 HPGD (0.56) TP53GAAMAPT
SCHEMBL6751301 0.77 MRGPRX4 (0.55) MAOBAPPNPC1RAB9ASMPD1
SCHEMBL6850661 0.74 MAOB (0.49) MAOBAPPNPC1RAB9ATDP1
SCHEMBL791922 0.72 MAOB (0.72) MAOBAPPNPC1RAB9ATDP1
SCHEMBL11955055 0.72 CYP2A6 (0.46) TP53MAPT
SCHEMBL6751659 0.71 SMPD1 (0.51) MAOBAPPNPC1RAB9ASMPD1
SCHEMBL4029474 0.71 NPC1 (0.57) MAOBAPPNPC1RAB9ATDP1
SCHEMBL791569 0.70 MAOB (1.00) MAOBAPPMRGPRX4
SCHEMBL18429793 0.70 APP (1.00) MAOBAPPNPC1RAB9ATDP1
SCHEMBL6751316 0.70 ERBB2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058265-A1 COMPOUND LIBRARIES OF 2,3-SUBSTITUTED PYRAZINE DERIVATIVES CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed