SCHEMBL6769332

SCHEMBL6769332

COc1ccc(CCCC(=O)c2ccc(CCC(C)(N)CO)s2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ALOX5 P09917 2/20 0.43
TRPV1 Q8NER1 1/20 0.43
TP53 P04637 1/20 0.41
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
ALDH1A1 P00352 1/20 0.39
F2RL1 P55085 1/20 0.39
S1PR4 O95977 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
MAPT P10636 1/20 0.38
PLAAT3 P53816 1/20 0.38
PLAAT5 Q96KN8 1/20 0.38
PLAAT2 Q9NWW9 1/20 0.38
PLAAT4 Q9UL19 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166232 0.97 HDAC4 (0.41) HDAC4HDAC6ALOX5TRPV1TP53
SCHEMBL5167475 0.89 MAPT (0.40) HDAC4HDAC6TRPV1TP53ALDH1A1
SCHEMBL6770520 0.88 S1PR1 (0.44) CASP3CASP7ALDH1A1S1PR4S1PR1
SCHEMBL5168391 0.87 POLB (0.40) HDAC4HDAC6TP53ALDH1A1S1PR1
SCHEMBL385258 0.86 TDP1 (0.43) HDAC4HDAC6TRPV1TP53CASP3
SCHEMBL6768979 0.86 NAMPT (0.41) TRPV1PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL5166925 0.86 S1PR1 (0.43) ALDH1A1S1PR4S1PR1S1PR3HPGD
SCHEMBL5168050 0.85 HDAC1 (0.47) HDAC6
SCHEMBL5167470 0.84 POLB (0.43) ALDH1A1S1PR4S1PR1S1PR3MAPT
SCHEMBL5169197 0.84 POLB (0.45) ALDH1A1S1PR4S1PR1S1PR3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723745-B2 PREVENTION OR TREATMENT OF AUTOIMMUNE DISEASE IN WARM BLOODED ANIMAL SANKYO COMPANY, LIMITED (JP) 2004-04-20 US claimed