SCHEMBL6770058

SCHEMBL6770058

CN1C(=O)CC(C)(C)c2cc(C(=O)C=Cc3ccc(C(=O)O)cc3)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
PTPN1 P18031 1/20 0.46
PTPN12 Q05209 1/20 0.46
PTPN22 Q9Y2R2 1/20 0.46
RARA P10276 9/20 0.46
RARB P10826 8/20 0.46
RARG P13631 8/20 0.46
RXRA P19793 3/20 0.46
STAT3 P40763 1/20 0.46
TP53 P04637 2/20 0.44
CYP3A4 P08684 2/20 0.44
BLM P54132 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HSD17B10 Q99714 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6770057 1.00 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6769121 0.90 HDAC1 (0.50) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6769123 0.90 HDAC1 (0.50) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL9593493 0.84 HDAC1 (0.56) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL4430921 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6765666 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6770031 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6765664 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL4424612 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6771219 0.83 RARB (0.45) HDAC3HDAC4HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6683092-B1 BREAST AND/OR PROSTATE CANCER ALLERGAN, INC. 2004-01-27 US disclosed