SCHEMBL6774737

SCHEMBL6774737

CC(C)(C)c1ccc(C(=O)Nc2ccsc2C(=O)Nc2cccc(C(=N)N)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK9 Q9NPC2 1/20 0.55
NR1H4 Q96RI1 9/20 0.53
KCNK3 O14649 1/20 0.51
PPARG P37231 3/20 0.50
PPARD Q03181 1/20 0.50
GPBAR1 Q8TDU6 1/20 0.50
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 2/20 0.49
RAB9A P51151 2/20 0.49
KMT2A Q03164 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
PLAU P00749 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6541293 0.99 KCNK9 (0.54) KCNK9NR1H4KCNK3PPARGPPARD
SCHEMBL12131818 0.83 F10 (0.53)
SCHEMBL10178439 0.81 F10 (0.43) KCNK9KCNK3PLAU
SCHEMBL6542489 0.81 NR1H4 (0.69) KCNK9NR1H4KCNK3MEN1ALDH1A1
SCHEMBL890957 0.81 F10 (0.60)
Hydrochloric Acid SCHEMBL6542009 0.81 NR1H4 (0.78) KCNK9NR1H4PPARGPPARDSMN1; SMN2
Hydrochloric Acid SCHEMBL6542404 0.80 CA1 (0.48) KCNK9NR1H4KCNK3PPARGPPARD
SCHEMBL6541256 0.77 KCNK9 (0.45) KCNK9NR1H4KCNK3PPARGPPARD
SCHEMBL6541251 0.77 KCNK9 (0.45) KCNK9NR1H4KCNK3PPARGPPARD
SCHEMBL13762080 0.77 KCNK9 (0.76) KCNK9NR1H4KCNK3PPARGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677369-B2 CARBOXIMIDAMIDE DERIVATIVE ANTICOAGULANTS INHIBIT FACTOR XA ELI LILLY AND COMPANY 2004-01-13 US claimed