SCHEMBL6780990

SCHEMBL6780990

CCOC(=O)CCN(C(=O)c1ccc2c(c1)nc(CNc1ccc(C#N)cc1OC)n2C)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F2 P00734 19/20 0.55
NQO2 P16083 1/20 0.54
NR1I2 O75469 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
SLC6A2 P23975 1/20 0.47
AGTR1 P30556 1/20 0.47
SLC6A3 Q01959 1/20 0.47
SCN5A Q14524 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6781433 0.92 F2 (0.56) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL6775238 0.91 F2 (0.56) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL7653930 0.91 NQO2 (0.67) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL6781845 0.89 NQO2 (0.65) F2NQO2NR1I2ADORA3SLC6A2
Hydrochloric Acid SCHEMBL6780913 0.88 F2 (0.69) F2NQO2
SCHEMBL6780877 0.85 F2 (0.60) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL6780096 0.84 NQO2 (0.60) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL506730 0.83 F2 (0.68) F2NQO2
SCHEMBL6785308 0.82 F2 (0.59) F2NQO2NR1I2ADORA3SLC6A2
SCHEMBL6781239 0.82 F2 (0.57) F2NQO2NR1I2ADORA3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6710055-B2 INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBO QUINOLINE-8-SULFONYLAMINO)-INDOLE BOEHRINGER INGELHEIM PHARMA GMBH & CO., KG (DE) 2004-03-23 US disclosed
US-6469039-B1 BENZIMIDAZOLES; THROMBIN- INHIBITING ACTIVITY AND THE EFFECT OF EXTENDING THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-10-22 US disclosed
US-6414008-B1 CYNAO- OR AMIDINE-SUBSTITUTED BENZIMIDAZOLES, BENOTHIAZOLES, OR BENZOXAZOLES; 2-(N-(4-AMIDINOPHENYL)AMINOMETHYL)BENZOTHIAZOLES; 2-((4-CYANOPHENYL)OXYMETHYL)IMIDAZOL(4,5-B)PYRIDINES; ANTITHROMBOTICS BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-07-02 US disclosed
US-6087380-A ANTITHROMBOTIC BENZIMIDAZOLES; ANTICOAGULANTS; 2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-BENZIMIDAZOL-5-YL-CARBOXYLIC ACIDS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-07-11 US disclosed