SCHEMBL6786783

SCHEMBL6786783

NC(=O)c1cccc2nc([C@H]3CC[C@H](C(=O)O)CC3)[nH]c12

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.50
PARP2 Q9UGN5 4/20 0.43
HTR2B P41595 1/20 0.42
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6783911 1.00 PARP1 (0.50) PARP1PARP2HTR2BADORA1
SCHEMBL6786430 0.88 PARP1 (0.50) PARP1PARP2HTR2B
SCHEMBL6782750 0.87 PARP1 (0.52) PARP1PARP2
SCHEMBL6778530 0.87 PARP1 (0.52) PARP1PARP2
SCHEMBL5074338 0.87 PARP1 (0.52) PARP1PARP2
SCHEMBL5072053 0.86 PARP1 (0.54) PARP1PARP2
SCHEMBL6781769 0.86 PARP1 (0.43) PARP1PARP2
SCHEMBL5619953 0.85 PARP1 (0.65) PARP1PARP2
SCHEMBL5077310 0.84 PBK (0.49) PARP1PARP2ADORA1
SCHEMBL5072056 0.84 PARP1 (0.71) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737421-B1 4-CARBOXYAMIDO SUBSTITUTED; NEURODEGENERATIVE DISEASES; NEURONAL DAMAGE ABBOTT GMBH & CO. KG (DE) 2004-05-18 US disclosed