SCHEMBL6788951

SCHEMBL6788951

O=c1[nH]nc(Cl)c(Cl)c1Cl

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TYMP P19971 2/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 2/20 0.31
ALDH1A1 P00352 1/20 0.31
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25072482 0.77
SCHEMBL8789178 0.74 HCAR2 (0.30) TYMPKMT2A
SCHEMBL25307884 0.69 DYRK1A (0.35) TYMPKMT2A
SCHEMBL29194141 0.67
SCHEMBL19668561 0.66 AR (0.34) AR
SCHEMBL599352 0.64 NPSR1 (0.57) POLBALDH1A1AR
SCHEMBL22164629 0.64 TYMP (0.35) TYMP
SCHEMBL2361036 0.64 TYMP (0.43) TYMPKMT2AALDH1A1AR
SCHEMBL9015978 0.64 AR (0.33) AR
SCHEMBL24687302 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6800758-B1 REACTING 4-(3-HALOPROPYLAMINO)-5- CHLORO-3(2H)-PYRIDAZINONE WITH N-METHYL- HOMOVERATRYLAMINE IN PRESENCE OF ACID BINDING AGENT AND DIPOLAR APROTIC SOLVENT EGIS GYOGYSZERGYAR RT. (HU) 2004-10-05 US disclosed
EP-0275997-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTAGONISTIC AGENT AGAINST SRS-A CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-12-23 EP disclosed
US-5011839-A Antagonists to slow reacting substance of anaphylaxis NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1991-04-30 US disclosed
US-4978665-A ANTIALLERGENS NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1990-12-18 US disclosed
EP-0376079-A1 3(2H)pyridazinones, processes for their preparation and antagonistic agent against SRS-A NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1990-07-04 EP disclosed
EP-0275997-A1 3(2H)pyridazinone, process for its preparation and antagonistic agent against SRS-A containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1988-07-27 EP disclosed