SCHEMBL6794181

SCHEMBL6794181

COCCN(C)CCCCC(=O)Nc1cccc(-c2n[nH]c(=O)c3ccccc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
ROCK1 Q13464 7/20 0.46
ROCK2 O75116 5/20 0.46
AURKA O14965 2/20 0.43
AURKB Q96GD4 2/20 0.43
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 2/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
BLM P54132 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
MAP4K4 O95819 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6786521 0.99 PARP1 (0.46) PARP1ROCK1ROCK2AURKAAURKB
SCHEMBL6786869 0.92 PARP1 (0.47) PARP1ROCK1ROCK2AURKAAURKB
Hydrochloric Acid SCHEMBL6792542 0.91 PARP1 (0.46) PARP1ROCK1ROCK2AURKAAURKB
SCHEMBL6783127 0.90 PARP1 (0.48) PARP1ROCK1ROCK2AURKAKDM4E
SCHEMBL6785898 0.90 PARP1 (0.53) PARP1ROCK1ROCK2AURKAAURKB
SCHEMBL6794194 0.90 PARP1 (0.47) PARP1ROCK1ROCK2AURKAAURKB
Hydrochloric Acid SCHEMBL6793382 0.89 PARP1 (0.48) PARP1ROCK1ROCK2AURKAKDM4E
Hydrochloric Acid SCHEMBL6788164 0.89 PARP1 (0.52) PARP1ROCK1ROCK2AURKAAURKB
SCHEMBL6792571 0.89 PARP1 (0.52) PARP1ROCK1ROCK2AURKAKDM4E
Hydrochloric Acid SCHEMBL6782482 0.89 PARP1 (0.47) PARP1ROCK1ROCK2AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677333-B1 ANTIISCHEMIC AGENTS; BRAIN, CARDIOVASCULAR, MUSCULAR, AND GASTROINTESTINAL DISORDERS; ANALGESICS, ANTIDIABETIC AGENTS; RETROVIRUS SENSITIZERS; ALZHEIMER*S DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2004-01-13 US claimed
EP-1148053-A1 2H-PHTHALAZIN-1-ONE DERIVATIVES AND DRUGS COMPRISING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-24 EP claimed