SCHEMBL679934

SCHEMBL679934

CS(=O)(=O)NC(=O)c1ccc(Oc2ccccc2)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.57
PNLIP P16233 2/20 0.49
MRGPRX4 Q96LA9 1/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
BCL2L1 Q07817 1/20 0.46
MCL1 Q07820 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679375 0.90 SCN9A (0.58) SCN9APNLIP
SCHEMBL679029 0.88 SCN9A (0.56) SCN9A
SCHEMBL680835 0.88 SCN9A (0.61) SCN9A
SCHEMBL680892 0.88 SCN9A (0.58) SCN9AMRGPRX4
SCHEMBL679751 0.88 SCN9A (0.58) SCN9A
SCHEMBL680538 0.88 SCN9A (0.53) SCN9AMRGPRX4
SCHEMBL366587 0.88 SCN9A (0.56) SCN9A
SCHEMBL16319549 0.87 SCN9A (0.58) SCN9ABCL2L1MCL1
SCHEMBL680190 0.87 SCN9A (0.55) SCN9AMRGPRX4
SCHEMBL16319475 0.86 SCN9A (0.62) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 13/4885PNLIP 4284/4885MRGPRX4 344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.