SCHEMBL6806014

SCHEMBL6806014

CN(C)CCCN(C)c1ccc(-c2nc3c(C(N)=O)cccc3[nH]2)cn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.63
MAP4K4 O95819 2/20 0.59
PIM1 P11309 2/20 0.59
PIM3 Q86V86 2/20 0.59
AURKB Q96GD4 2/20 0.59
CLK4 Q9HAZ1 2/20 0.59
STK17A Q9UEE5 2/20 0.59
MAP4K5 Q9Y4K4 2/20 0.59
DYRK3 O43781 1/20 0.59
RPS6KB1 P23443 1/20 0.59
CSNK2A1 P68400 1/20 0.59
PKN2 Q16513 1/20 0.59
BRSK1 Q8TDC3 1/20 0.59
HIPK2 Q9H2X6 1/20 0.59
MKNK2 Q9HBH9 1/20 0.59
DHODH Q02127 3/20 0.59
CHEK1 O14757 1/20 0.56
LCK P06239 1/20 0.56
CSF1R P07333 1/20 0.56
PHKG2 P15735 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806654 0.94 PARP1 (0.66) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6803442 0.87 CHEK1 (0.68) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6591145 0.86 PARP1 (0.46) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6806881 0.85 AURKB (0.61) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6805128 0.85 AURKB (0.66) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6806027 0.84 CHEK2 (0.43) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6810671 0.83 AURKB (0.63) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6806488 0.83 PARP1 (0.61) PARP1PIM1PIM3AURKBCLK4
SCHEMBL7134204 0.83 PARP1 (0.67) PARP1MAP4K4PIM1PIM3AURKB
SCHEMBL6807295 0.83 AURKB (0.63) PARP1MAP4K4PIM1PIM3AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed