SCHEMBL681202

SCHEMBL681202

C=C(C(C)C)[C@H](CN[C@@H]1CCNC1)c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
KCNH2 Q12809 2/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A3 Q01959 2/20 0.36
SSTR4 P31391 1/20 0.35
HTR3A P46098 1/20 0.35
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681297 1.00 SLC6A2 (0.38) SLC6A2SLC6A4KCNH2CYP2D6SLC6A3
SCHEMBL680936 0.88 SLC6A2 (0.40) SLC6A2SLC6A4KCNH2CYP2D6SSTR4
SCHEMBL680723 0.88 SLC6A2 (0.40) SLC6A2SLC6A4KCNH2CYP2D6SSTR4
SCHEMBL681566 0.86 MEN1 (0.40) CYP2D6GAAHPGDSMN1; SMN2
SCHEMBL684480 0.85 SLC6A4 (0.40) SLC6A2SLC6A4KCNH2SLC6A3SSTR4
SCHEMBL684494 0.85 SLC6A4 (0.40) SLC6A2SLC6A4KCNH2SLC6A3SSTR4
SCHEMBL2738619 0.83 CHEK1 (0.38)
SCHEMBL2738616 0.83 CHEK1 (0.38)
SCHEMBL680141 0.83 AKT3 (0.45) CYP2D6GAAHPGDSMN1; SMN2
SCHEMBL680114 0.81 BRD4 (0.42) GAAHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed