SCHEMBL6814766

SCHEMBL6814766

COCCCCn1c(=O)c(C)nc2c(-c3ccc(OC)cc3Cl)ccnc21

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
STK4 Q13043 1/20 0.43
STK3 Q13188 1/20 0.43
SIK2 Q9H0K1 1/20 0.43
STK26 Q9P289 1/20 0.43
STK24 Q9Y6E0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6817809 0.91 PDE4B (0.47)
SCHEMBL6818381 0.90 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6814314 0.90
SCHEMBL6817702 0.90
SCHEMBL6819066 0.87
SCHEMBL6814575 0.86
SCHEMBL6818786 0.86 STK4 (0.42) STK4STK3SIK2STK26STK24
SCHEMBL6817739 0.86 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6818951 0.85
SCHEMBL6822425 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO claimed
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed