SCHEMBL6818645

SCHEMBL6818645

CC(Nc1nccc(-c2cc(F)c(N(C)C)cc2Cl)c1N)C1CC1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.37
SOS1 Q07889 8/20 0.36
IDH2 P48735 2/20 0.34
IDO1 P14902 2/20 0.32
BCL6 P41182 1/20 0.32
MDM2 Q00987 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6082791 1.00 IDH1 (0.37) IDH1SOS1IDH2IDO1BCL6
SCHEMBL6082490 0.96 MDM2 (0.35) IDH1SOS1IDH2BCL6MDM2
SCHEMBL6081890 0.87 SOS1 (0.39) IDH1SOS1IDH2IDO1
SCHEMBL6082255 0.84 IDH1 (0.36) IDH1SOS1IDH2IDO1BCL6
SCHEMBL6082249 0.84 IDH1 (0.36) IDH1SOS1IDH2IDO1BCL6
SCHEMBL6082565 0.82 KDM4E (0.34)
SCHEMBL6082474 0.80 MDM2 (0.35) IDH1SOS1IDH2IDO1BCL6
SCHEMBL6082481 0.80 MDM2 (0.35) IDH1SOS1IDH2IDO1BCL6
SCHEMBL6818651 0.79 BRD4 (0.34)
SCHEMBL6814612 0.77 BCHE (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004031189-A1 PYRIDINO AND PYRIMIDINO PYRAZINONES FOR TREATMENT OF ANXIETY AND DEPRESSION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2004-04-15 WO disclosed