SCHEMBL6822671

SCHEMBL6822671

CC(C)(O)c1cnc(C(=Cc2cccc(-c3cc(C(C)(C)C#N)cc4cccnc34)c2)c2ccccc2S(C)(=O)=O)s1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 16/20 0.59
PDE4B Q07343 16/20 0.59
PDE4C Q08493 16/20 0.59
PDE4D Q08499 16/20 0.59
CYP2C9 P11712 5/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822670 1.00 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4030234 0.89 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4030231 0.89 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027814 0.79 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4025227 0.76 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4025224 0.76 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027365 0.74 PDE4A (0.90) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027369 0.74 PDE4A (0.90) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4028925 0.74 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4031232 0.74 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6740666-B2 FOR THERAPY OF ASTHMA, CHRONIC BRONCHITIS, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, EOSINOPHILIC GRANULOMA, PSORIASIS; SEPTIC SHOCK, ULCERATIVE COLITIS, CROHN'S DISEASE, REPERFUSION INJURY OF THE MYOCARDIUM AND BRAIN, INFLAMMATION MERCK & CO., INC. 2004-05-25 US disclosed