SCHEMBL6823595

SCHEMBL6823595

COc1ccc2c(-c3ccc(OCCN(C)C)cc3)c(Oc3ccc(Cl)cc3Cl)c(=O)oc2c1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.61
CYP19A1 P11511 1/20 0.45
CSF1R P07333 2/20 0.45
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
SIGMAR1 Q99720 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6819971 0.91 ESR1 (0.63) ESR1CYP19A1CSF1RCA1CA2
SCHEMBL6823204 0.90 ESR1 (0.72) ESR1CYP19A1CSF1RCA1CA2
SCHEMBL6823324 0.86 ESR1 (0.77) ESR1CSF1RCA1CA2SIGMAR1
SCHEMBL6823503 0.84 NPC1 (0.49) ESR1CYP19A1CA1CA2KDM4E
SCHEMBL6922082 0.83 ESR1 (0.73) ESR1CSF1RSIGMAR1BCHEACHE
SCHEMBL6922106 0.83 ESR1 (0.72) ESR1CSF1RSIGMAR1BCHEACHE
SCHEMBL6823220 0.80 ESR1 (0.77) ESR1CSF1RALDH1A1
SCHEMBL6823739 0.80 ESR1 (0.67) ESR1CYP19A1SIGMAR1BCHEACHE
SCHEMBL6921522 0.78 ESR1 (0.56) ESR1CSF1RSIGMAR1
SCHEMBL8951798 0.75 ESR1 (0.53) ESR1CYP19A1CSF1RCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004069820-A1 COUMARIN DERIVATIVES HAVING AN AFFINITY FOR OESTROGEN RECEPTORS, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME B.F.B. ETUDES ET RECHERCHES EXPERIMENTALES (FR) 2004-08-19 WO disclosed