SCHEMBL6825637

SCHEMBL6825637

CC(C)(C)C(=S)c1nc2c(N)ncnc2n1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ENTPD1 P49961 3/20 0.69
TRPM2 O94759 1/20 0.60
RNASEL Q05823 1/20 0.59
P2RY1 P47900 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16805436 0.86 ENTPD1 (0.77) ENTPD1TRPM2RNASELP2RY1
SCHEMBL18852609 0.86 ENTPD1 (0.77) ENTPD1TRPM2RNASELP2RY1
SCHEMBL21283084 0.86 ENTPD1 (0.77) ENTPD1TRPM2RNASELP2RY1
SCHEMBL18858917 0.86 ENTPD1 (0.77) ENTPD1TRPM2RNASELP2RY1
SCHEMBL636535 0.85 ENTPD1 (0.75) ENTPD1TRPM2P2RY1
SCHEMBL636536 0.85 ENTPD1 (0.75) ENTPD1TRPM2P2RY1
SCHEMBL29398104 0.84 ENTPD1 (0.74) ENTPD1TRPM2P2RY1
SCHEMBL12932272 0.84 ENTPD1 (0.76) ENTPD1TRPM2P2RY1
SCHEMBL374912 0.84 ENTPD1 (0.73) ENTPD1TRPM2P2RY1
SCHEMBL15082696 0.84 ENTPD1 (0.73) ENTPD1TRPM2P2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043955-A1 C8-substituted purine nucleotide analogs and their use as inhibitors of nucleoside triphosphate diphosphohydrolases BEAUDOIN ADRIEN R (CA) 2004-03-04 US disclosed
US-6617439-B1 Adenine with a thioether substituent; use as enzyme inhibitors; modulates conversion into nucleosides BAR-ILAN UNIVERSITY (IL) 2003-09-09 US disclosed