SCHEMBL6826366

SCHEMBL6826366

COc1ccc2[nH]c3c(N4CCN(CCc5ccc(F)c(F)c5)CC4)ncnc3c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 16/20 1.00
CYP3A4 P08684 7/20 0.87
ABCB1 P08183 2/20 0.68
HRH4 Q9H3N8 2/20 0.67
KDM4E B2RXH2 2/20 0.62
ALDH1A1 P00352 2/20 0.62
LMNA P02545 2/20 0.62
MAPT P10636 2/20 0.62
HIF1A Q16665 2/20 0.62
STAT6 P42226 1/20 0.62
HTT P42858 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
IDE P14735 1/20 0.58
HPGD P15428 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7135303 0.93 ABCC1 (1.00) ABCC1CYP3A4ABCB1HRH4KDM4E
SCHEMBL6923887 0.90 ABCC1 (0.81) ABCC1CYP3A4ABCB1HRH4KDM4E
SCHEMBL6920584 0.86 ABCC1 (0.77) ABCC1CYP3A4ABCB1KDM4EALDH1A1
SCHEMBL6826593 0.86 ABCC1 (0.77) ABCC1CYP3A4ABCB1KDM4EALDH1A1
SCHEMBL6827154 0.86 ABCC1 (1.00) ABCC1CYP3A4ABCB1KDM4EALDH1A1
SCHEMBL6828902 0.83 ABCC1 (1.00) ABCC1CYP3A4ABCB1ABCG2
SCHEMBL6918220 0.83 ABCC1 (0.86) ABCC1CYP3A4ABCB1KDM4EALDH1A1
SCHEMBL6826699 0.83 ABCC1 (0.81) ABCC1CYP3A4ABCB1KDM4EALDH1A1
SCHEMBL6826415 0.83 ABCC1 (1.00) ABCC1CYP3A4ABCB1ABCG2
SCHEMBL6922901 0.82 ABCC1 (0.82) ABCC1CYP3A4ABCB1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO claimed
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed