SCHEMBL6826440

SCHEMBL6826440

Cc1ccc(C(=O)c2ccc(O)c(-c3cc(N4CCOCC4)nc(N)n3)c2)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.55
CDK2 P24941 4/20 0.55
RAF1 P04049 4/20 0.45
BRAF P15056 3/20 0.45
HPGD P15428 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
MAPT P10636 2/20 0.40
AKT1 P31749 2/20 0.39
PIK3CA P42336 2/20 0.39
MTOR P42345 2/20 0.39
PDPK1 O15530 1/20 0.38
PRKDC P78527 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6823630 0.94 CDK1 (0.49) CDK1CDK2RAF1BRAF
SCHEMBL6918875 0.90 CDK1 (0.55) CDK1CDK2
SCHEMBL6825113 0.89 CDK1 (0.44) CDK1CDK2RAF1BRAF
SCHEMBL6820798 0.83 CDK1 (0.40) CDK1CDK2RAF1BRAF
SCHEMBL7068093 0.83 RAF1 (0.45) CDK1CDK2RAF1BRAFHPGD
SCHEMBL6820704 0.82 CDK1 (0.59) CDK1CDK2HPGDALDH1A1SMN1; SMN2
SCHEMBL6824190 0.82 MAPK14 (0.43) CDK1CDK2ALDH1A1SMN1; SMN2
SCHEMBL6824305 0.81 MAPK14 (0.48) CDK1CDK2HPGDALDH1A1SMN1; SMN2
SCHEMBL6824361 0.81 MAPK14 (0.40) CDK1CDK2HPGDALDH1A1LMNA
SCHEMBL6826271 0.81 KDM4E (0.41) CDK1CDK2ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO claimed
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed