SCHEMBL6826635

SCHEMBL6826635

CC(C)Oc1nc(C2CC2)nc(OC(C)C)c1Br

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.35
PDE8B O95263 1/20 0.33
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
CSNK2A1 P68400 1/20 0.32
CHRM3 P20309 3/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320750 0.77 CCNA2 (0.36) PDE10A
SCHEMBL11443735 0.75 PDE10A (0.39) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL6826203 0.73 DHODH (0.32) PDE10A
SCHEMBL6826298 0.71 PDE4D (0.32) PDE4D
SCHEMBL6826154 0.71 PDE10A (0.41) PDE10APDE8BCHRM3PDE4APDE4B
SCHEMBL6340021 0.67 CNR2 (0.31)
SCHEMBL11444512 0.67 PDE10A (0.33) PDE10A
SCHEMBL6341152 0.66 PDE10A (0.36) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL5321886 0.65 CSNK2A2 (0.35) CSNK2A2CSNK2BCSNK2A1
SCHEMBL6336289 0.65 EDNRB (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111000-A2 PIPERIDYL DERIVATIVES AND THEIR USE AS TACHYKININ ANTAGONISTS ASTELLAS PHARMA INC. (JP) 2004-12-23 WO disclosed