SCHEMBL6829633

SCHEMBL6829633

COc1ccc([N+](=O)[O-])cc1C1CCNC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.54
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
SLC6A3 Q01959 1/20 0.54
HTR2A P28223 3/20 0.52
HTR2C P28335 2/20 0.52
CHRNB4 P30926 3/20 0.51
CHRNA3 P32297 3/20 0.51
HTT P42858 1/20 0.49
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
PDE4B Q07343 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6785307 0.92 HTR2C (0.54) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
Bicarbonate SCHEMBL6716536 0.86 HTR2C (0.48) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
Bicarbonate SCHEMBL6716542 0.86 HTR2C (0.48) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
Bicarbonate SCHEMBL6716532 0.85 CYP2D6 (0.47) CYP2D6SLC6A2SLC6A4SLC6A3HTR2C
SCHEMBL1531299 0.84 TDP1 (0.57) CHRNB4CHRNA3HTTTDP1ALDH1A1
SCHEMBL22609007 0.80 CHRNB4 (0.55) SLC6A2SLC6A4SLC6A3CHRNB4CHRNA3
SCHEMBL7898068 0.77 HTR2C (0.60) HTR2AHTR2CPDE4B
Hydrochloric Acid SCHEMBL23326197 0.76 HTR2C (0.58) HTR2AHTR2CPDE4B
Hydrochloric Acid SCHEMBL29775341 0.76 HTR2C (0.58) HTR2AHTR2CPDE4B
SCHEMBL18952921 0.75 CHRNB4 (0.50) CYP2D6SLC6A2SLC6A4SLC6A3CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004010943-A2 SUBSTITUTED BENZANILIDES AS MODULATORS OF THE CCR5 RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2004-02-05 WO disclosed
EP-0380063-B1 1,2-CYCLOHEXYLAMINOARYL AMIDES USEFUL AS ANALGESIC AGENTS WARNER-LAMBERT COMPANY (US) 1993-07-21 EP disclosed
US-5019588-A Nonhabit-forming analgeiscs WARNER-LAMBERT COMPANY (US) 1991-05-28 US disclosed
EP-0380063-A1 1,2-cyclohexylaminoaryl amides useful as analgesic agents WARNER-LAMBERT COMPANY (US) 1990-08-01 EP disclosed
US-4906655-A Novel 1,2-cyclohexylaminoaryl amides useful as analgesic agents WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed