SCHEMBL6832198

SCHEMBL6832198

COc1ccc(CS(=O)(=O)C(C)(C)[C@@H](N)C(=O)N2CC(F)CC2C#N)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 1.00
FAP Q12884 9/20 0.81
DPP7 Q9UHL4 3/20 0.79
DPP8 Q6V1X1 1/20 0.68
DPP9 Q86TI2 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6860819 1.00 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
SCHEMBL3165078 1.00 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
SCHEMBL5987446 1.00 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
Hydrochloric Acid SCHEMBL356162 0.99 DPP4 (0.98) DPP4FAPDPP7DPP8DPP9
Hydrochloric Acid SCHEMBL295498 0.99 DPP4 (0.98) DPP4FAPDPP7DPP8DPP9
SCHEMBL3160316 0.90 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
SCHEMBL3159890 0.90 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
SCHEMBL8353910 0.90 DPP4 (1.00) DPP4FAPDPP7DPP8DPP9
SCHEMBL3156933 0.90 DPP4 (1.00) DPP4FAPDPP7
Hydrochloric Acid SCHEMBL3259953 0.89 DPP4 (0.98) DPP4FAPDPP7DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092128-A1 ANHYDROUS CRYSTALLINE FORMS OF (2S, 4S)-1-{(2R)-2-AMINO-3-‘4-METHOXYBENZYL)SULFONYL!-3-METHYLBUTANOYL}-4-FLUOROPYRROLINDINE-2-CARBONITRILE SMITHKLINE BEECHAM CORPORATION (US) 2004-10-28 WO claimed
WO-2004092128-A1 ANHYDROUS CRYSTALLINE FORMS OF (2S, 4S)-1-{(2R)-2-AMINO-3-‘4-METHOXYBENZYL)SULFONYL!-3-METHYLBUTANOYL}-4-FLUOROPYRROLINDINE-2-CARBONITRILE SMITHKLINE BEECHAM CORPORATION (US) 2004-10-28 WO disclosed