SCHEMBL6833474

SCHEMBL6833474

CNc1nc(NC2CCCCC2N(C(=O)C(F)(F)F)c2ccc(F)c(F)c2)ncc1C

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.42
SYK P43405 8/20 0.38
ADRA2A P08913 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
HTR2B P41595 1/20 0.38
PTK2 Q05397 6/20 0.36
PTK2B Q14289 4/20 0.35
FGFR4 P22455 1/20 0.35
MAPK3 P27361 3/20 0.34
MAPK1 P28482 3/20 0.34
KCNH2 Q12809 3/20 0.34
AURKB Q96GD4 3/20 0.34
GP6 Q9HCN6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6455574 0.84 MCHR1 (0.51) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6456487 0.79 MCHR1 (0.49) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6464501 0.77 MCHR1 (0.45) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6456500 0.75 MCHR1 (0.47) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6456465 0.71 MCHR1 (0.47) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6459587 0.70 MCHR1 (0.52) MCHR1ADRA2AADRA1AHRH1HTR2B
SCHEMBL6461142 0.70 MCHR1 (0.48) MCHR1SYKADRA2AADRA1AHRH1
SCHEMBL6455417 0.70 MCHR1 (0.56) MCHR1ADRA2AADRA1AHRH1HTR2B
Trifluoroacetic Acid SCHEMBL6833473 0.69 MCHR1 (0.67) MCHR1ADRA2AADRA1AHRH1HTR2B
Trifluoroacetic Acid SCHEMBL6455569 0.69 MCHR1 (0.67) MCHR1ADRA2AADRA1AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087669-A1 NOVEL QUINOLINE, TETRAHYDROQUINAZOLINE, AND PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO. LTD. (JP) 2004-10-14 WO disclosed