SCHEMBL6847895

SCHEMBL6847895

[CH2]C#Cc1ccc(-c2nccc(OC)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.38
CLK4 Q9HAZ1 4/20 0.38
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP4B1 P13584 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP3A5 P20815 1/20 0.36
CYP2A7 P20853 1/20 0.36
CYP3A7 P24462 1/20 0.36
CYP2F1 P24903 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852660 0.81 NPC1 (0.38) NPC1MEN1KMT2AMAPTALDH1A1
SCHEMBL6854125 0.80 MEN1 (0.38) NPC1MEN1KMT2AMAPTALDH1A1
SCHEMBL7031581 0.79 NPC1 (0.45) NPC1MEN1KMT2AMAPTALDH1A1
SCHEMBL7031587 0.77 MEN1 (0.53) NPC1MEN1KMT2AMAPTALDH1A1
Ammonia Solution, Strong SCHEMBL28862501 0.76 MEN1 (0.51) NPC1MEN1KMT2AMAPTALDH1A1
SCHEMBL21051576 0.76 MEN1 (0.64) NPC1MEN1KMT2AMAPTCLK4
SCHEMBL2130866 0.76 MEN1 (0.51) NPC1MEN1KMT2AMAPTCLK4
SCHEMBL28020382 0.75 NPC1 (0.60) NPC1MEN1KMT2AMAPTCLK4
SCHEMBL15483941 0.75 KMT2A (0.50) NPC1MEN1KMT2AMAPTALDH1A1
SCHEMBL29524578 0.75 KMT2A (0.50) NPC1MEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed