SCHEMBL6851624

SCHEMBL6851624

Clc1cccc(Cl)c1-c1cc2c3c(c1)[C@H]1CNCC[C@H]1CN3CCC2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 14/20 0.40
HTR2B P41595 7/20 0.40
HTR2A P28223 7/20 0.40
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HTR6 P50406 1/20 0.32
KCNH2 Q12809 1/20 0.31
CHRNB2 P17787 2/20 0.30
CHRNB4 P30926 2/20 0.30
CHRNA3 P32297 2/20 0.30
CHRNA4 P43681 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3136180 1.00 HTR2C (0.40) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL13268789 1.00 HTR2C (0.40) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL3136412 0.85 HTR2C (0.42) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL13270187 0.85 HTR2C (0.42) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL13270124 0.85 HTR2C (0.43) HTR2CHTR2BHTR2AKMT2AKCNH2
SCHEMBL3138083 0.85 HTR2C (0.43) HTR2CHTR2BHTR2AKMT2AKCNH2
SCHEMBL5415878 0.81 HTR2C (0.55) HTR2CHTR2BHTR2AKCNH2
SCHEMBL3140380 0.80 HTR2C (0.57) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL13270210 0.80 HTR2C (0.57) HTR2CHTR2BHTR2AMAPTKDM4E
SCHEMBL3127409 0.80 PTPN11 (0.39) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6777406-B2 SUCH AS PYRIDO(3,2,1-IJ)PYRROLO(3,4-C)QUINOLIN-8-ONE DERI-VATIVES; CENTRAL NERVOUS SYSTEM DISORDERS; GASTROINTESTINAL DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-08-17 US disclosed