SCHEMBL6851642

SCHEMBL6851642

O=C(O)c1c(CN2CCN(C(=O)CCN3CCOCC3)CC2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 13/20 0.54
TACR2 P21452 10/20 0.54
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KCNH2 Q12809 3/20 0.47
HTR7 P34969 3/20 0.46
HTR1A P08908 1/20 0.46
OPRM1 P35372 3/20 0.45
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5459898 0.91 TACR2 (0.53) TACR3TACR2KCNH2HTR7OPRM1
SCHEMBL5462467 0.90 TACR3 (0.55) TACR3TACR2KCNH2OPRM1
SCHEMBL4903021 0.89 TACR3 (0.63) TACR3TACR2ALDH1A1KCNH2OPRM1
Hydrochloric Acid SCHEMBL7683491 0.88 TACR3 (0.62) TACR3TACR2ALDH1A1KCNH2OPRM1
SCHEMBL5461424 0.86 TACR2 (0.53) TACR3TACR2ALDH1A1KCNH2OPRM1
SCHEMBL5450782 0.82 TACR3 (0.51) TACR3TACR2ALDH1A1SMN1; SMN2KCNH2
SCHEMBL6853329 0.81 TACR2 (0.57) TACR3TACR2ALDH1A1KCNH2OPRM1
SCHEMBL6853049 0.81 TACR3 (0.58) TACR3TACR2KCNH2OPRM1TSHR
SCHEMBL6853022 0.81 TACR3 (0.51) TACR3TACR2KCNH2OPRM1
SCHEMBL5455427 0.81 TACR2 (0.53) TACR3TACR2KCNH2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US claimed
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US disclosed