SCHEMBL6852463

SCHEMBL6852463

C=C1c2ccccc2C(=O)N1C[C@H]1CO1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
ALDH1A1 P00352 5/20 0.46
DHFR P00374 1/20 0.44
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.40
HBB P68871 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MIF P14174 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
GLS O94925 1/20 0.39
MEN1 O00255 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14410468 1.00 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL29570568 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL767566 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL29567211 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL29402853 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL38819 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL78821 0.88 CYP2C9 (0.68) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR
SCHEMBL6914233 0.82 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL13651922 0.76 CYP1A2 (0.66) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL17983178 0.75 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19ALDH1A1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005028-A2 METHOD FOR PREPARING (S)-5-CHLORO-N-((3-(4-(5,6-DIHYDRO-4H-1,2,4-OXADIAZIN-3-YL)PHENYL)-2-OXOOXAZOLIDIN-5-YL)METHYL)THIOPHENE-2-CARBOXAMIDE DERIVATIVES LEGOCHEM BIOSCIENCE LTD. (KR) 2011-01-13 WO disclosed