SCHEMBL6857591

SCHEMBL6857591

Nc1nc(-c2ccc(F)cc2)c2c(n1)-c1c(cccc1-c1ccccc1)C2=O

nearest known ligand 0.65

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.65
ADORA2A P29274 19/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1881088 0.92 ADORA2A (0.77) ADORA1ADORA2A
SCHEMBL1880456 0.90 ADORA2A (0.60) ADORA1ADORA2A
SCHEMBL1882224 0.86 ADORA2A (0.63) ADORA1ADORA2A
SCHEMBL1881060 0.86 ADORA1 (0.57) ADORA1ADORA2A
SCHEMBL1878234 0.86 ADORA2A (0.57) ADORA1ADORA2A
SCHEMBL1879453 0.85 ADORA2A (0.61) ADORA1ADORA2A
SCHEMBL1758596 0.85 ADORA1 (0.59) ADORA1ADORA2A
SCHEMBL12660096 0.84 ADORA2A (0.70) ADORA1ADORA2A
SCHEMBL1881399 0.84 ADORA2A (0.50) ADORA1ADORA2A
SCHEMBL1881942 0.83 ADORA2A (0.65) ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011053509-A1 ARYL SUBSTITUTED ARYLINDENOPYRIMIDINES AND THEIR USE AS HIGHLY SELECTIVE ADENOSINE A2A RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed