SCHEMBL6858614

SCHEMBL6858614

CC(NC(=O)C=Cc1ccc(Br)cc1)C1=COC=C(C2=CC=CCC2)O1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
TDP1 Q9NUW8 1/20 0.35
GPR183 P32249 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 2/20 0.34
KDM4E B2RXH2 1/20 0.34
RAB9A P51151 1/20 0.34
KCNQ2 O43526 2/20 0.33
CYP3A4 P08684 2/20 0.33
KCNQ3 O43525 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP2C9 P11712 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
RECQL P46063 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6646805 0.84 KCNQ2 (0.36) LMNATDP1ALDH1A1CYP1A2KDM4E
SCHEMBL3210780 0.71 AKR1B1 (0.47)
SCHEMBL5171573 0.68 KMT2A (0.35) LMNARAB9AMEN1KMT2A
SCHEMBL3729102 0.68
SCHEMBL4831678 0.67
SCHEMBL8194241 0.66
SCHEMBL3619674 0.66
SCHEMBL2177347 0.65 TNIK (0.33)
SCHEMBL3103877 0.64
SCHEMBL5909441 0.64 SNCA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831080-B2 E.g., 3-(2-fluorophenyl)-N-(1-(3-morpholin-4-yl)phenyl)-propyl)acrylamide; disorders responsive to opening of KCNQ potassium channels; analgesics; migraine, bipolar disorders, anticonvulsants, antiepileptic, anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY 2004-12-14 US disclosed