SCHEMBL6861992

SCHEMBL6861992

COc1ccc(CC(C)(C)NCC(O)COc2ccc(NS(C)(=O)=O)cc2C#N)cc1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASR P41180 18/20 0.68
ADRB2 P07550 8/20 0.68
CYP2D6 P10635 8/20 0.68
SLC6A2 P23975 7/20 0.68
SLC6A4 P31645 7/20 0.68
SLC6A3 Q01959 7/20 0.68
KCNH2 Q12809 7/20 0.68
ADRB3 P13945 4/20 0.68
ADRB1 P08588 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861982 1.00 CASR (0.68) CASRADRB2CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6862969 0.99 CASR (0.67) CASRADRB2CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6862981 0.99 CASR (0.67) CASRADRB2CYP2D6SLC6A2SLC6A4
SCHEMBL6857917 0.89 CASR (0.62) CASRADRB2CYP2D6SLC6A2SLC6A4
SCHEMBL6857912 0.89 CASR (0.62) CASRADRB2CYP2D6SLC6A2SLC6A4
SCHEMBL6863615 0.88 CASR (0.73) CASRADRB2CYP2D6SLC6A2SLC6A4
SCHEMBL6863624 0.88 CASR (0.73) CASRADRB2CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6863062 0.88 CASR (0.61) CASRADRB2CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6863826 0.87 CASR (0.72) CASRADRB2CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL6863834 0.87 CASR (0.72) CASRADRB2CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP claimed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US claimed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP claimed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO claimed
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed