SCHEMBL6862358

SCHEMBL6862358

CN1CCN(c2cc(C(=O)N(C)Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c(-c3ccccc3Cl)cn2)CC1

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.72
TACR3 P29371 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637377 0.93 TACR1 (0.83) TACR1TACR3
Hydrochloric Acid SCHEMBL905337 0.92 TACR1 (0.81) TACR1TACR3
SCHEMBL4119209 0.89 TACR1 (0.73) TACR1
SCHEMBL4111340 0.88 TACR1 (0.70) TACR1
SCHEMBL4114128 0.87 TACR1 (0.69) TACR1
Hydrochloric Acid SCHEMBL5743257 0.87 TACR1 (0.68) TACR1
SCHEMBL4117598 0.84 TACR1 (0.67) TACR1
SCHEMBL905330 0.84 TACR1 (1.00) TACR1
SCHEMBL29467378 0.84 TACR1 (1.00) TACR1
SCHEMBL4131710 0.83 TACR1 (0.82) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157005-B1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2004-10-20 EP claimed
EP-1157005-A1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-28 EP claimed
US-6225316-B1 GOOD AFFINITY TO THE NK-1 RECEPTOR. HOFFMANN-LA ROCHE INC. 2001-05-01 US claimed
WO-2000050401-A1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-08-31 WO claimed
EP-1157005-B1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2004-10-20 EP disclosed
EP-1157005-A1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-28 EP disclosed
US-6225316-B1 GOOD AFFINITY TO THE NK-1 RECEPTOR. HOFFMANN-LA ROCHE INC. 2001-05-01 US disclosed
WO-2000050401-A1 3-PHENYLPYRIDINE DERIVATIVES AND THEIR USE AS NK-1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-08-31 WO disclosed