SCHEMBL6862797

SCHEMBL6862797

CC(C)c1ccc(COc2ccc(CC(=O)O)cc2Cl)cc1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.67
PPARD Q03181 3/20 0.56
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
HPGD P15428 1/20 0.54
MRGPRX4 Q96LA9 4/20 0.52
RXRA P19793 3/20 0.50
RXRB P28702 3/20 0.50
RXRG P48443 2/20 0.50
ADRB3 P13945 4/20 0.48
CA2 P00918 1/20 0.48
FFAR1 O14842 2/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
XBP1 P17861 1/20 0.47
HTT P42858 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PPARA Q07869 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11473142 0.88 PPARD (0.55) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11470785 0.86 PPARD (0.58) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL29394534 0.86 PPARD (0.60) PPARDNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL3950358 0.86 PPARD (0.60) PPARDNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11460459 0.86 PPARD (0.53) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11460782 0.85 PPARD (0.55) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11460696 0.85 PPARD (0.55) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11465700 0.85 PPARD (0.52) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11462250 0.84 PPARD (0.57) PDK2PPARDNPC1RAB9ASMN1; SMN2
SCHEMBL11462528 0.83 MRGPRX4 (0.62) PDK2PPARDNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040058425-A1 Crystal structure PFIZER INC. 2004-03-25 US disclosed
EP-1247860-A1 Crystal structure of pyruvate dehydrogenase kinase 2 (PDHK-2) and use thereof in methods for identifying and designing new ligands Pfizer Limited (GB) 2002-10-09 EP disclosed
US-4221919-A Antiinflammatory substituted phenylacetic acids SPOFA, UNITED PHARMACEUTICAL WORKS (CS) 1980-09-09 US disclosed