SCHEMBL6863079

SCHEMBL6863079

Cc1ccsc1-c1nc2cc(C(=O)N(C(C)C)C(C)C)cc(N)n2n1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.42
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MCOLN3 Q8TDD5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867491 0.89 ADORA2A (0.47) ADORA2A
SCHEMBL6870499 0.85 ADORA2A (0.59) ADORA2AHPGD
SCHEMBL6871231 0.85 ADORA2A (0.45) ADORA2AHPGDNPSR1
SCHEMBL6867741 0.84 ADORA2A (0.46) ADORA2AHPGD
SCHEMBL6871350 0.82 ADORA2A (0.41) ADORA2A
SCHEMBL6871970 0.81 ADORA2A (0.43) ADORA2AHPGD
SCHEMBL6867399 0.79 ADORA2A (0.67) ADORA2AHPGD
SCHEMBL6869056 0.78 ADORA2A (0.66) ADORA2AHPGD
SCHEMBL6870464 0.77 ADORA2A (0.42) ADORA2A
SCHEMBL6870459 0.77 ADORA2A (0.43) ADORA2AHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed