SCHEMBL6863261

SCHEMBL6863261

Cc1ccccc1-c1ccccc1OC(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.67
CETP P11597 1/20 0.53
GPBAR1 Q8TDU6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872781 0.83 TACR1 (0.74) TACR1GPBAR1
SCHEMBL5779738 0.82 TACR1 (0.59) TACR1GPBAR1
SCHEMBL5781646 0.81 TACR1 (0.54) TACR1GPBAR1
SCHEMBL6872779 0.80 TACR1 (1.00) TACR1
SCHEMBL6871449 0.79 TACR1 (0.55) TACR1GPBAR1
SCHEMBL6016603 0.79 TACR1 (0.50) TACR1CETPGPBAR1
SCHEMBL5763724 0.78 TACR1 (0.61) TACR1GPBAR1
SCHEMBL6016671 0.78 TACR1 (0.49) TACR1CETPGPBAR1
SCHEMBL5781165 0.77 TACR1 (0.49) TACR1GPBAR1
SCHEMBL8785556 0.77 TACR1 (0.73) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171419-B1 BIPHENYL DERIVATIVES AS ANTAGONISTS OF THE NEUROKININE-1 RECEPTOR HOFFMANN LA ROCHE (CH) 2004-12-29 EP claimed