SCHEMBL6863435

SCHEMBL6863435

Nc1cc(C(=O)N2CC=CCC2)cc2nc(-c3nccs3)nn12

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.51
ABL1 P00519 3/20 0.36
BCR P11274 3/20 0.36
HPGD P15428 1/20 0.36
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870494 0.93 ADORA2A (0.53) ADORA2AABL1BCRHPGDADORA2B
SCHEMBL6863814 0.86 ADORA2A (0.67) ADORA2AABL1BCRHPGD
SCHEMBL6863682 0.85 ADORA2A (0.66) ADORA2AABL1BCRHPGD
SCHEMBL6870030 0.85 ADORA2A (0.66) ADORA2AABL1BCRHPGD
SCHEMBL6863267 0.85 ADORA2A (0.66) ADORA2AABL1BCRHPGD
SCHEMBL6870405 0.85 ADORA2A (0.60) ADORA2AABL1BCRHPGD
SCHEMBL6871629 0.83 ADORA2A (0.53) ADORA2AABL1BCRHPGDADORA2B
SCHEMBL6870280 0.82 ADORA2A (0.53) ADORA2AABL1BCRHPGD
SCHEMBL6872125 0.81 ADORA2A (0.50) ADORA2AHPGD
SCHEMBL6871877 0.80 ADORA2A (0.48) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed