SCHEMBL6864449

SCHEMBL6864449

COc1cc2nccc(Oc3ccc(NC(=O)Nc4cc(C)on4)cc3)c2cc1OC

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 19/20 0.76
KDR P35968 19/20 0.76
FLT1 P17948 2/20 0.75
EPHB2 P29323 2/20 0.75
FLT4 P35916 2/20 0.75
RIPK2 O43353 1/20 0.75
STK10 O94804 1/20 0.75
ABL1 P00519 1/20 0.75
LCK P06239 1/20 0.75
LYN P07948 1/20 0.75
RET P07949 1/20 0.75
MET P08581 1/20 0.75
PDGFRB P09619 1/20 0.75
KIT P10721 1/20 0.75
BCR P11274 1/20 0.75
FGFR1 P11362 1/20 0.75
SRC P12931 1/20 0.75
MAPK3 P27361 1/20 0.75
HTR2A P28223 1/20 0.75
MAPK1 P28482 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21174284 0.99 PDGFRA (0.74) PDGFRAKDRFLT1EPHB2FLT4
SCHEMBL1873986 0.96 PDGFRA (0.70) PDGFRAKDRFLT1EPHB2FLT4
SCHEMBL29973354 0.89 PDGFRA (0.95) PDGFRAKDR
SCHEMBL27081475 0.89 PDGFRA (0.95) PDGFRAKDR
SCHEMBL21174250 0.89 PDGFRA (0.73) PDGFRAKDR
SCHEMBL6376965 0.87 FLT3 (0.79) PDGFRAKDRFLT1EPHB2FLT4
SCHEMBL3931065 0.86 PDGFRA (1.00) PDGFRAKDR
SCHEMBL5651032 0.86 KDR (0.81) PDGFRAKDRFLT1EPHB2FLT4
Tivozanib SCHEMBL172883 0.86 KDR (1.00) PDGFRAKDRFLT1EPHB2FLT4
Hydrochloric Acid SCHEMBL5653983 0.86 FLT3 (0.78) PDGFRAKDRFLT1EPHB2FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040242603-A1 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus proliferator receptor and medicinal composition containing the same KIRIN HOLDINGS KABUSHIKI KAISHA (JP) 2004-12-02 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040242603-A1 Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus proliferator receptor and medicinal composition containing the same NR1H2, NR1H3, NR1H4 PDGFRA 1364/4885KDR 1874/4885FLT1 3370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.