E2Mate

E2Mate

SCHEMBL6866434

C[C@]12CCC3c4ccc(OS(N)(=O)=O)cc4CCC3C1CC[C@H]2O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 9/20 1.00
ABCC1 P33527 1/20 0.83
ABCC4 O15439 1/20 0.83
KDM4E B2RXH2 1/20 0.81
CA1 P00915 2/20 0.76
CA2 P00918 2/20 0.76
CA9 Q16790 2/20 0.76
LMNA P02545 4/20 0.75
HSD17B10 Q99714 4/20 0.75
ESR1 P03372 5/20 0.73
PGR P06401 2/20 0.73
AR P10275 2/20 0.73
SLC6A3 Q01959 2/20 0.73
SMN1; SMN2 Q16637 2/20 0.73
ADORA3 P0DMS8 1/20 0.73
CHRM1 P11229 1/20 0.73
TBXA2R P21731 1/20 0.73
ADRA1A P35348 1/20 0.73
OPRM1 P35372 1/20 0.73
ATM Q13315 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
E2Mate SCHEMBL19272474 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL628174 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL5165269 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL5980613 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL29924099 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL5151234 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL10070158 1.00 STS (1.00) STSABCC1ABCC4KDM4ECA1
Emate SCHEMBL7164522 0.93 STS (0.86) STSABCC1ABCC4KDM4ECA1
E2Mate SCHEMBL15940838 0.91 STS (0.83) STSABCC1ABCC4KDM4ECA1
SCHEMBL232796 0.91 ABCC4 (1.00) STSABCC1ABCC4KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775155-B1 ESTRA-1,3,5(10)-TRIENE DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING AG (DE) 2004-05-06 EP claimed
US-6080735-A SUITABLE FOR HORMONAL CONTRACEPTION AND CLIMACTERIC HORMONE REPLACEMENT THERAPY (HRT) AS WELL AS FOR TREATMENT OF GYNECOLOGICAL AND ANDROLOGICAL DISEASES JENAPHARM GMBH & CO. KG (DE) 2000-06-27 US claimed
EP-0775155-B1 ESTRA-1,3,5(10)-TRIENE DERIVATIVES, METHODS OF PREPARING SUCH COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING AG (DE) 2004-05-06 EP disclosed
US-6080735-A SUITABLE FOR HORMONAL CONTRACEPTION AND CLIMACTERIC HORMONE REPLACEMENT THERAPY (HRT) AS WELL AS FOR TREATMENT OF GYNECOLOGICAL AND ANDROLOGICAL DISEASES JENAPHARM GMBH & CO. KG (DE) 2000-06-27 US disclosed