SCHEMBL6869347

SCHEMBL6869347

Cc1cccc(Cl)c1NC(=O)N[C@H]1CC[C@@H](Nc2nc3c(c(N(C)C)n2)CCCC3)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.46
LCK P06239 4/20 0.45
MCHR1 Q99705 13/20 0.44
ADRA2A P08913 10/20 0.44
HRH1 P35367 5/20 0.44
HTR2B P41595 5/20 0.44
MAPK14 Q16539 2/20 0.43
ADRA1A P35348 2/20 0.42
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869351 1.00 EPHX1 (0.46) EPHX1LCKMCHR1ADRA2AHRH1
SCHEMBL6879572 0.95 MCHR1 (0.44) EPHX1LCKMCHR1ADRA2AHRH1
SCHEMBL6879578 0.95 MCHR1 (0.44) EPHX1LCKMCHR1ADRA2AHRH1
SCHEMBL6879285 0.93 EPHX1 (0.53) EPHX1LCKMCHR1ADRA2AHRH1
SCHEMBL6879288 0.93 EPHX1 (0.53) EPHX1LCKMCHR1ADRA2AHRH1
SCHEMBL6463027 0.89 MCHR1 (0.46) LCKMCHR1ADRA2AHRH1HTR2B
SCHEMBL6463030 0.89 MCHR1 (0.46) LCKMCHR1ADRA2AHRH1HTR2B
SCHEMBL6872737 0.88 SMN1; SMN2 (0.56) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6872741 0.88 SMN1; SMN2 (0.56) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6462544 0.88 EPHX1 (0.45) EPHX1MCHR1ADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed