SCHEMBL6870243

SCHEMBL6870243

CC1C=CC(C)N1C(=O)c1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.44
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863575 0.88 ADORA2A (0.45) ADORA2AADORA2BADORA1
SCHEMBL6863363 0.87 ADORA2A (0.47) ADORA2AADORA2BADORA1
SCHEMBL6863359 0.87 ADORA2A (0.47) ADORA2AADORA2BADORA1
SCHEMBL6870280 0.82 ADORA2A (0.53) ADORA2A
SCHEMBL6871877 0.82 ADORA2A (0.48) ADORA2A
SCHEMBL6863122 0.82 ADORA2A (0.45) ADORA2AADORA2BADORA1
SCHEMBL6867753 0.81 ADORA2A (0.61) ADORA2A
SCHEMBL6870494 0.81 ADORA2A (0.53) ADORA2AADORA2BADORA1
SCHEMBL6863814 0.81 ADORA2A (0.67) ADORA2A
SCHEMBL6867359 0.80 ADORA2A (0.62) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed